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BI 7189
CAS No. 1883429-32-0
BI 7189 ( BI7189 )
产品货号. M12928 CAS No. 1883429-32-0
BI 7189 is a highly selective bromodomains of BRD9 and BRD7 inhibitor with IC50<50 nM for BRD9.
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| 规格 | 价格/人民币 | 库存 | 数量 |
| 100MG | 获取报价 | 有现货 |
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| 200MG | 获取报价 | 有现货 |
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| 500MG | 获取报价 | 有现货 |
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| 1G | 获取报价 | 有现货 |
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生物学信息
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产品名称BI 7189
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注意事项本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
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产品简述BI 7189 is a highly selective bromodomains of BRD9 and BRD7 inhibitor with IC50<50 nM for BRD9.
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产品描述BI 7189 is a highly selective bromodomains of BRD9 and BRD7 inhibitor with IC50<50 nM for BRD9, displays >1,000 fold selectivity over the bromodomains of BRD4; suppresses the proliferation of AML cells.
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同义词BI7189
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通路Chromatin/Epigenetic
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靶点Bromodomain
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受体Bromodomain
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研究领域——
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适应症——
化学信息
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CAS Number1883429-32-0
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分子量330.43
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分子式C19H26N2O3
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纯度>98% (HPLC)
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溶解度——
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SMILES——
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化学全称5-[4-[(dimethylamino)methyl]-3,5-dimethoxyphenyl]-1,3,6-trimethylpyridin-2-one
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1. Hohmann AF, et al. Nat Chem Biol. 2016 Sep;12(9):672-9.
2. Pérez-Salvia M, et al. Epigenetics. 2017 May 4;12(5):323-339.
2. Pérez-Salvia M, et al. Epigenetics. 2017 May 4;12(5):323-339.
产品手册
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